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Ligand 4-[4-(aminosulfonyl)phenyl]-1-(2'-acetamido-2'-deoxy'-3',4',6'-tri-O-acetyl-beta-D-glucopyranosyl)-1H-1,2,3-triazole

Basic Ligand Information

Molecular Structure

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Roles as Enzyme Ligand

Inhibitor in Enzyme-catalyzed Reactions (1 result)

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Show Inhibitors (1 entry)

EC NUMBER

COMMENTARY

LITERATURE

ENZYME 3D STRUCTURE

4.2.1.1

-

699426

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Enzyme Kinetic Parameters

K_i Value (3 results)

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Show KI Value (3 entries)

EC NUMBER

KI VALUE [MM]

KI VALUE MAXIMUM [MM]

COMMENTARY

LITERATURE

4.2.1.1

0.000101

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isozyme CA IX, in 10 mM HEPES (pH 7.5), 0.1 M NaClO4, at 20°C

699426

4.2.1.1

0.00044

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isozyme CA II, in 10 mM HEPES (pH 7.5), 0.1 M NaClO4, at 20°C

699426

4.2.1.1

0.005

-

isozyme CA I, in 10 mM HEPES (pH 7.5), 0.1 M NaClO4, at 20°C

699426

4.2.1.1

3 entries

References & Links

Literature References (1)

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Show Reference (1 entry)

BRENDA REFERENCE ID

PUBMED ID

TITLE

YEAR

AUTHORS

JOURNAL

VOLUME

PAGES

699426

18307288

Inhibition of carbonic anhydrases with glycosyltriazole benzene sulfonamides

2008

Wilkinson, B.L.; Innocenti, A.; Vullo, D.; Supuran, C.T.; Poulsen, S.A.

J. Med. Chem.

51

1945-1953

Links to other databases for 4-[4-(aminosulfonyl)phenyl]-1-(2'-acetamido-2'-deoxy'-3',4',6'-tri-O-acetyl-beta-D-glucopyranosyl)-1H-1,2,3-triazole

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Show Links (1 entry)

ChEBI

PubChem

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